APIs Intermediates CAS No. | ||
Resmetirom | 6-(4-amino-2,6-dichlorophenoxy)-4- isopropylpyridazin-3(2H)-one | 920509-28-0 |
3,5-dichloro-4-((6-chloro-5-isopropylpyridazin-3- yl)oxy)aniline | 920509-27-9 | |
N-Cyanoacetylurethane | 6629-04-5 | |
Abrocitinib | Benzyl(1s,3s)-3-(methyl(7-tosyl-7H-pyrrolo[2,3- d]pyrimidin-4-yl)amino)cyclobutyl)carbamate | 1622903-41-6 |
4-Chloropyrrolo[2,3-d]pyrimidine | 3680-69-1 | |
Asenapine Maleate | 1-Bromo-2-bromomethyl-4-chlorobenzene | 66192-24-3 |
Apremilast | 3-Acetamidophthalic anhydride | 6296-53-3 |
3-Ethoxy-4-methoxy-alpha-[(methylsulfonyl)methyl]- benzenemethanamine | 253168-94-4 | |
3-Ethoxy-4-methoxybenzonitrile | 60758-86-3 | |
Apalutamide | 5-Amino-3-(trifluoromethyl)pyridine-2-carbonitrile | 573762-62-6 |
Vibegron | (6S)-4,6,7,8-tetrahydro-4-0xo-Pyrrolo[1,2- a]pyriMidine-6-carboxylic acid | 1190392-22-3 |
Vortioxetine Hydrobromide | 1-Bromo-2-iodobenzene | 583-55-1 |
2,4-Dimethylbenzenethiol | 13616-82-5 | |
Vericiguat | 2-chloro-5-fluoronicotinamide | 113237-20-0 |
5-fluoro-1H-pyrazolo[3,4-b]pyridin-3-amine | 1034667-22-5 | |
Valbenazine | 6,7-Dimethoxy-3,4-dihydroisoquinoline hydrochloride | 20232-39-7 |
3-(N,N-Dimethylaminomethyl)-5-methyl-2-hexanone | 91342-74-4 | |
Vonoprazan | 3-Pyridinesulfonyl chloride | 16133-25-8 |
5-(2-Fluoropheny)-1H-pyrrole-3-carboxaldehyde | 881674-56-2 | |
Tofacitinib Citrate | N-Methyl-N-[(3R,4R)-4-methyl-1-(phenylmethyl)-3- piperidinyl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine | 477600-73-0 |
(2R,3R)-2,3-Bis[(4-methylbenzoyl)oxy]butanedioic acid compd.with (3R,4R)-N,4-dimethyl-1-(phenylmethyl)- 3-piperidinamine | 477600-71-8 | |
4-Chloropyrrolo[2,3-d]pyrimidine | 3680-69-1 | |
Suvorexant | (R)-5-chloro-2-(5-methyl-1,4-diazepan-1- yl)benzo[d]oxazole | 1266975-27-2 |
5-methyl-2-(2H-1,2,3-triazol-2-yl)benzoicacid | 956317-36-5 | |
Siponimod | 1-(3-ethyl-4-(hydroxymethyl)phenyl)ethan-1-one | 1378888-43-7 |
Sacubitril | (2R,4S)-5-(biphenyl-4-y)-4-[(tert-butoxycarbonyl) amino]-2-methylpentanoic acid | 1012341-50-2 |
Selexipag | 5-Chloro-2,3-diphenylpyrazine | 41270-66-0 |
4-[(5,6-Diphenylpyraziny)(1-methylethyl)amino]-1- butanol | 475086-75-0 | |
Ruxolitinib | -(1-Ethoxyethyl)-1H-pyrazole-4-boronic acid pinacol ester | 1029716-44-6 |
4-Chloropyrrolo[2,3-d]pyrimidine | 3680-69-1 | |
Prasugrel | 5,6,7,7a-Tetrahydrothieno[3,2-c]pyridinone Hydrochloride | 115473-15-9 |
2-Bromo-2-(2-fluorophenyl)-1-cyclopropylethanone | 204205-33-4 | |
Perampanel Hydrate | 5-Bromo-2-methoxypyridine | 13472-85-0 |
2-Bromopyridine | 109-04-6 | |
Pemafibrate | 3-(4-methoxyphenoxy)propan-1-amine | 100841-00-7 |
Oxcarbazepine | 10-Methoxyiminostilbene | 4698/11/7 |
Opicapone | 2,5-Dichloro-4,6-dimethylnicotinonitrile | 91591-63-8 |
Mirogabalin | (1R,5S)-3-Ethylbicyclo[3.2.0]hept-3-en-6-one | 1235479-61-4 |
2-Aminothiazol-4-acetic acid | 29676-71-9 | |
Macitentan | 4,6-Dichloro-5-(4-bromophenyl)pyrimidine | 146533-41-7 |
N-Propyl-sulfamide potassium salt | 1393813-41-6 | |
5-Bromo-2-chloropyrimidine | 32779-36-5 | |
Lurasidone Hydrochloride | (1R,2R)-1,2-cyclohexanedimethanol | 65376-05-8 |
Cis-5-Norborene钬摇xo-2,3-dicarboxylic anhydride | 2746-19-2 | |
Lemborexant | 2,4-Dimethyl-5-pyrimidinol | 412003-95-3 |
(1 R,2S)-2-(3-fluorophenyl)-2-((p- tosyloxy)methyl)cyclopropyl)methyl acetate | 1450904-92-3 | |
Ivabradine hydrochloride | (1S)-4,5-Dimethoxy-1- [(methylamino)methyl]benzocyclobutane hudrochlorida | 866783-13-3 |
1,3-Dihydro-3-(3-iodopropyl)-7,8-dimethoxy-2H-3- benzazepin-2-one | 148870-57-9 | |
Guanfacine hydrochloride | 2,6-Dichlorophenylacetic acid | 6575-24-2 |
Evocalcet | Ethyl4-bromophenylacetate | 14062-25-0 |
(S)-N-((R)-1-(naphthalen-1-y)ethyl)pyrrolidin-3-amine | 870966-25-9 | |
Esaxerenone | 1H-Pyrrole-3-carboxylic acid,4-methyl-5-[2- (trifluoromethyl)phenyl]-,ethyl ester | 1631030-76-6 |
Enzalutamide | 4-Isothiocyanato-2-(trifluoromethyl)benzonitrile | 143782-23-4 |
N-[3-Fluoro-4-[(methylamino)carbonyl]phenyl]-2- methylalanine | 1289942-66-0 | |
Eltrombopag Olamine | 3'-Amino-2'-hydroxy-[1,1'-biphenyl]-3-carboxylic acid | 376592-93-7 |
3-Methyl-1-(3,4-dimethylphenyl)-2-pyrazolin-5-one | 18048-64-1 | |
Elobixibat hydrate | (R)--[N-(t-butoxycarbonylmethyl) carbamoyl]benzylamine | 439088-74-1 |
7-bromo-3,3-dibutyl-8-methoxy-2,3- dihydrobenzo[b][1,4]thiazepine-4(5H)-one | 439089-27-7 | |
4-Methylenepiperidine hydrochloride | 144230-50-2 | |
2-Aminothiazol-4-acetic acid | 29676-71-9 | |
Macitentan | 4,6-Dichloro-5-(4-bromophenyl)pyrimidine | 146533-41-7 |
N-Propyl-sulfamide potassium salt | 1393813-41-6 | |
5-Bromo-2-chloropyrimidine | 32779-36-5 | |
Lurasidone Hydrochloride | (1R,2R)-1,2-cyclohexanedimethanol | 65376-05-8 |
Cis-5-Norborenexo-2,3-dicarboxylic anhydride | 2746-19-2 | |
Lemborexant | 2,4-Dimethyl-5-pyrimidinol | 412003-95-3 |
(1 R,2S)-2-(3-fluorophenyl)-2-((p- tosyloxy)methyl)cyclopropyl)methyl acetate | 1450904-92-3 | |
Ivabradine hydrochloride | (1S)-4,5-Dimethoxy-1- [(methylamino)methyl]benzocyclobutane hudrochlorida | 866783-13-3 |
1,3-Dihydro-3-(3-iodopropyl)-7,8-dimethoxy-2H-3- benzazepin-2-one | 148870-57-9 | |
Guanfacine hydrochloride | 2,6-Dichlorophenylacetic acid | 6575-24-2 |
Evocalcet | Ethyl4-bromophenylacetate | 14062-25-0 |
(S)-N-((R)-1-(naphthalen-1-y)ethyl)pyrrolidin-3-amine | 870966-25-9 | |
Esaxerenone | 1H-Pyrrole-3-carboxylic acid,4-methyl-5-[2- (trifluoromethyl)phenyl]-,ethyl ester | 1631030-76-6 |
Enzalutamide | 4-Isothiocyanato-2-(trifluoromethyl)benzonitrile | 143782-23-4 |
N-[3-Fluoro-4-[(methylamino)carbonyl]phenyl]-2- methylalanine | 1289942-66-0 | |
Eltrombopag Olamine | 3'-Amino-2'-hydroxy-[1,1'-biphenyl]-3-carboxylic acid | 376592-93-7 |
3-Methyl-1-(3,4-dimethylphenyl)-2-pyrazolin-5-one | 18048-64-1 | |
Elobixibat hydrate | (R)--[N-(t-butoxycarbonylmethyl) carbamoyl]benzylamine | 439088-74-1 |
7-bromo-3,3-dibutyl-8-methoxy-2,3- dihydrobenzo[b][1,4]thiazepine-4(5H)-one | 439089-27-7 | |
4-Methylenepiperidine hydrochloride | 144230-50-2 | |
1-Chloroethyl cyclohexyl carbonate | 99464-83-2 | |
Ezetimibe | (3R,4S)-4-[4-(Benzyloxy)phenyl]-1-(4-fluoropheny)-3- [3-(4-fluoropheny)-3-oxopropyl]azetidin-2-one | 190595-65-4 |
Deucravacitinib Sofosbuvir | ethyl 4,6-dihydroxypyridazine-3-carboxylate | 1352925-63-3 |
METHYL-D3-AMINE HYDROCHLORIDE | 7436-22-8 | |
2-methoxy-3-(1-methyl-1H-1,2,4-triazol-3-yl)aniline | 1609394-10-6 | |
N-[(S)-(2,3,4,5,6-Penta fluorophenoxy)phenoxy phosphinyl]-L-alanine 1-methylethyl ester | 1334513-02-8 | |
(2'R)-2'-Deoxy-2'-fluoro-2'-methyluridine) | 863329-66-2 | |
Dolutegravir | (3R)-3-Amino-1-butanol | 61477-40-5 |
Methyl 4-methoxyacetoacetate | 41051-15-4 | |
2,4-Difluorobenzylamine | 72235-52-0 | |
1-(2,2-Dimethoxyethyl)-1,4-dihydro-3-methoxy-4- oxo-2,5-pyridinedicarboxylicacid 2-methyl ester | 1335210-23-5 | |
(1R,2S)-rel-2-(3,4-Difluoro phenyl)cyclopropanamine hydrochloride | 1156491-10-9 | |
4,6-Dichloro-2-propyl thiopyrimidine-5-amine | 145783-15-9 | |
2-(3aR,4S,6R,6aS)-6-Amino-2,2-dimethyltetrahydro- 3aH-cyclopenta[d][1,3]dioxol-4-yloxy)ethanol L- tataric ncid | 376608-65-0 | |
Velpatasvir | (2S,4S)-2-[5-[1,11-Dihydro-2-[(2S,5S)-1-[(2S)-2-[( methoxycarbonyl)amino]-3-methyl-1-oxobutyl]-5- methyl-2-pyrrolidinyl][2]benzopyrano[4,3':6,7] naphth[1,2-d]imidazol-9-yl]-1H-imidazol-2-yl]-4- (methoxymethyl)-1-pyrrolidinecarboxylic acid 1,1- dimethylethyl ester | 1378391-45-7 |
Posaconazole | N'-((2S,3S)-2-(Benzyloxy)pentan-3-yl)formohydrazide oxalate | 1887197-42-3 |
2-[(1S,2S)-1-Ethyl-2-benzyloxypropyl]-2,4-dihydro-4- [4-[4-(4-hydroxyphenyl)-1-piperazinyl]phenyl]-3H- 1,2,4-triazol-3-one | 184177-83-1 | |
[S-(R',R')]-2,3-Bis (benzoyloxy)butanedioic acid compd.with [S-(R,R)]-[1-ethyl-2-(phenylmethoxy) propyl]hydrazine | 183871-36-5 | |
Valsartan/Sa cubitril | (2R,4S)-5-(Biphenyl-4-yl)-4-[(tert-butoxycarbonyl) amino]-2-methylpentanoic acid | 1012341-50-2 |
(2R,4S)-4-Amino-5-(biphenyl-4-yl)-2-methyl pentanoic acid ethyl ester hydrochloride | 149690-12-0 | |
Sacubitril hemicalcium salt | 1369773-39-6 | |
Venetoclax | Methyl 2-[(1H-pyrrolo[2,3-b]pyridin-5-yl)oxy]-4- fluoro benzoate | 1235865-75-4 |
1-((4'-chloro-5,5-dimethyl-3,4,5,6-tetrahydro-[1,1'- biphenyl]-2-yl)methyl)piperazine | 1228780-72-0 | |
Ibrutinib | (S)-1-Boc-3-hydroxy piperidine | 143900-44-1 |
3-(4-Phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-4- amine | 330786-24-8 | |
Acalabrutinib | [4-[(Pyridin-2-yl)carbamoyl]phenyl]boronic acid | 850568-25-1 |
(S)-Benzyl 2-(8-amino-1-bromoimidazo[1,5-a]pyrazin- 3-yl)pyrrolidine-1-carboxylate | 1420478-88-1 | |
N-(Pyridin-2-yl)-4-(4,4,5,5-tetramethyl-1,3,2- dioxaborolan-2-yl)benzamide | 1383385-64-5 | |
Upadacitinib | (3R,4S)-3-(2-Bromoacetyl)-4-ethyl-1- pyrrolidinecarboxylic acid phenylmethyl ester | 1428243-26-8 |
Tert-butyl 5-tosyl-5H-pyrrolo[2,3-b]pyrazin-2- ylcarbamate | 1201187-44-1 |
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